Compile Data Set for Download or QSAR
maximum 50k data
Found 5435 of ic50 data for polymerid = 354,3113,50001378,999,5864
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166892(CHEMBL3797772)
Affinity DataIC50:  0.0100nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166881(CHEMBL3798535)
Affinity DataIC50:  0.0100nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166880(CHEMBL3798487)
Affinity DataIC50:  0.0200nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50447747(CHEMBL3113272)
Affinity DataIC50:  0.0250nMAssay Description:Apparent inhibition of human FAAH expressed in CHOK1 cells using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166868(CHEMBL3797635)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166873(CHEMBL3800456)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166871(CHEMBL3797841)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166866(CHEMBL3798156)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50447748(CHEMBL3113271)
Affinity DataIC50:  0.0720nMAssay Description:Apparent inhibition of human FAAH expressed in CHOK1 cells using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166869(CHEMBL3799744)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50447745(CHEMBL3113274)
Affinity DataIC50:  0.0800nMAssay Description:Apparent inhibition of human FAAH expressed in CHOK1 cells using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166890(CHEMBL3797809)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50350535(CHEMBL1812722)
Affinity DataIC50:  0.0930nMAssay Description:Inhibition of FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50132714((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenesulfonyl f...)
Affinity DataIC50:  0.100nMAssay Description:Irreversible inhibition of fatty acid amide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50161525(1-(oxazolo[4,5-b]pyridin-2-yl)-9-phenylnonan-1-one...)
Affinity DataIC50:  0.100nMAssay Description:Inhibitory concentration of fatty acid amide hydrolase using FP-Rh radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
University Of California

Curated by ChEMBL
LigandPNGBDBM50132713(Arachidonic acid derivative | CHEMBL113262 | Methy...)
Affinity DataIC50:  0.100nMAssay Description:Inhibitory potency of Fatty-acid amide hydrolase with Mouse brain memebraneMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
University Of California

Curated by ChEMBL
LigandPNGBDBM50247048(CHEMBL462609 | methyl icosylphosphonofluoridate)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of FAAH-mediated [3H]anadamide hydrolysis in mouse brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50236330(CHEMBL4070196)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
University Of California

Curated by ChEMBL
LigandPNGBDBM50132714((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenesulfonyl f...)
Affinity DataIC50:  0.110nMAssay Description:Inhibitory potency of Fatty-acid amide hydrolase with Mouse brain memebraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166867(CHEMBL3798476)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Mus musculus (mouse))
University Of California

Curated by ChEMBL
LigandPNGBDBM50247052(2-Nonylsulfanyl-4H-benzo[1,3,2]dioxaphosphinine 2-...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of FAAH-mediated [3H]anadamide hydrolysis in mouse brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50309725(CHEMBL598764 | nicotinaldehyde O-4-(undecyloxy)phe...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166910(CHEMBL3798355)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50250852(CHEMBL4078217)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of human recombinant FAAH using arachidonoyl-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50447747(CHEMBL3113272)
Affinity DataIC50:  0.170nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166911(CHEMBL3799516)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50309712(4-fluorobenzaldehyde O-4-(nonyloxy)phenylcarbamoyl...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166891(CHEMBL3799008)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50166878(CHEMBL3800599)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM359728(US10435355, Example 12 | US9822068, 12 | [3-(3-car...)
Affinity DataIC50:  0.230nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM359728(US10435355, Example 12 | US9822068, 12 | [3-(3-car...)
Affinity DataIC50:  0.230nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50295654(CHEMBL559034 | Dodecylcarbamic acid 3-(1,2,3-thiad...)
Affinity DataIC50:  0.240nMAssay Description:Inhibition of FAAH in Wistar rat cerebral membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM26739(3-(3-carbamoylphenyl)phenyl N-cyclohexylcarbamate ...)
Affinity DataIC50:  0.240nMAssay Description:Inhibition of MBP-fused human recombinant FAAH with truncated N-terminal transmembrane domain expressed in Escherichia coli T7 using D-AMC substrate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50309701(CHEMBL597430 | benzaldehyde O-4-(nonyloxy)phenylca...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50309713(4-fluorobenzaldehyde O-4-(decyloxy)phenylcarbamoyl...)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50309711(4-fluorobenzaldehyde O-4-(octyloxy)phenylcarbamoyl...)
Affinity DataIC50:  0.270nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50447746(CHEMBL3113273)
Affinity DataIC50:  0.280nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50551026(CHEMBL4749527)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50434318(CHEMBL2386566)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of human FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50236334(CHEMBL4071240)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50437233(CHEMBL2402911)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Wistar rat brain FAAH using [3H]-ethanolamine as substrate preincubated for 20 mins followed by substrate addition by liquid scintillat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50161520(1-(oxazolo[4,5-b]pyridin-2-yl)-8-phenyloctan-1-one...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration of fatty acid amide hydrolase using FP-Rh radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM23316(7-phenyl-1-{pyrido[2,3-d][1,3]oxazol-2-yl}heptan-1...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration of fatty acid amide hydrolase using FP-Rh radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM23316(7-phenyl-1-{pyrido[2,3-d][1,3]oxazol-2-yl}heptan-1...)
Affinity DataIC50:  0.300nMAssay Description:Inhibitory concentration against Fatty-acid amide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM23316(7-phenyl-1-{pyrido[2,3-d][1,3]oxazol-2-yl}heptan-1...)
Affinity DataIC50:  0.316nMpH: 9.0 T: 2°CAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [3H]anandamide was evaluated by using rat brain homogenate preparations. [3H]Ethanola...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50132713(Arachidonic acid derivative | CHEMBL113262 | Methy...)
Affinity DataIC50:  0.330nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50419129(CHEMBL1830441)
Affinity DataIC50:  0.331nMAssay Description:Displacement of [3H]-anandamide from rat brain FAAH after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50132713(Arachidonic acid derivative | CHEMBL113262 | Methy...)
Affinity DataIC50:  0.331nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Assam University (A Central University)

Curated by ChEMBL
LigandPNGBDBM50447745(CHEMBL3113274)
Affinity DataIC50:  0.340nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
E.I. Du Pont De Nemours

Curated by ChEMBL
LigandPNGBDBM50309702(CHEMBL597431 | benzaldehyde O-4-(decyloxy)phenylca...)
Affinity DataIC50:  0.350nMAssay Description:Inhibition of human FAAH expressed in human H4 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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